P&T News: Jan/Feb 2000

Appropriate Use of Antibiotics: The Antibiotic Advisory Subcommittee and You

Dena M. Behm-Dillon, Pharm.D.
Peer Review Status: Internally Peer Reviewed by Antibiotic Advisory Subcommittee


Antibiotic therapy has become the focus of growing public attention because of concerns about microbial resistance and reduced patient safety seen with the inappropriate use of these important agents. The UIHC has taken significant steps to ensure that all antimicrobials are prescribed safely and in a manner to keep drug resistance to a minimum. The purposes of this article are to describe the Antibiotic Advisory Subcommittee and the Protocol Antibiotic Program, review UIHC-specific microbial susceptibility data, and discuss the appropriate use of several commonly ordered serum antibiotic levels.

The Antibiotic Advisory Subcommittee (AAS)
The AAS is composed of members drawn from a variety of disciplines. The co-chairs are from the Infectious Diseases service, and other members are from Pediatrics, Medical I.C.U., Surgical I.C.U., Obstetrics/Gynecology, Surgery, Microbiology, Pharmacy, and Epidemiology. The AAS is an advisory subcommittee to the Pharmacy and Therapeutics (P&T) Subcommittee. The P&T Subcommittee, in turn, reports directly to the Hospital Advisory Committee.

The AAS has three primary functions:

1. To analyze anti-infective use and microbial sensitivity patterns within the UIHC and provide recommendations as appropriate to the Pharmacy and Therapeutics Subcommittee.

2. To advise the Pharmacy and Therapeutics Subcommittee regarding the anti-infectives that should be stocked at UIHC.

3. To advise the Pharmacy and Therapeutics Subcommittee on whether a medication use evaluation should be conducted on the use of an anti-infective and to assist in criteria development.

 There are four steps which implement the primary functions of the AAS, each completed in collaboration with Pharmacy and Medical staffs. These include

1. Targeting specific drugs for appropriate dosing, susceptibility patterns, and safety issues, e.g. protocol antibiotics;

2. Development of criteria for antibiotic utilization proposals;

3. Implementation and monitoring the program; and

4. Review of results through data analysis and quarterly report review.

Protocol Antibiotic Program
Many of the objectives of the AAS are met through the Protocol Antibiotic Program. The program was implemented in 1992 as a collaborative effort of the AAS, the Pharmacy and Therapeutics Subcommittee, the Medication Use Evaluation Subcommittee, and the Medical Staff. The "protocol" classification includes those anti-infectives which have been approved for stock with the restriction they be used only according to specific criteria. The criteria can be obtained from the protocol forms which are in file boxes on each inpatient care unit.

The purposes of this program are to: prevent development of drug-resistant organisms through appropriate anti-infective selection and monitoring; pinpoint primary drug uses; and finally, monitor the success of strategies to control costs. This last step is conducted through prospective therapeutic drug monitoring by clinical pharmacists and a series of computer-generated reports. The reports describe purchasing, inventory, and drug utilization for inpatients, clinic patients, and the UIHC Ambulatory Care Pharmacies. They permit ongoing review by the AAS, Pharmacy and Therapeutics Subcommittee, and respective departments of drug products and quantities dispensed by pharmacy, drug expenses and susceptibility data for specific patient care units/clinical services, and changes in utilization over time. Feedback is provided through data analysis and quarterly report review. Quarterly reports are then distributed to all clinical departments for review and follow-up, as needed. The Protocol Antibiotic Program facilitates optimal patient care through promotion of appropriate prescribing, and it serves as a means of addressing concerns regarding microbial resistance.

Susceptibility Data

The "Guide to Choice of Antibiotic Therapy", published twice yearly by the UIHC, includes information provided by the Departments of Pathology (Medical Microbiology) and Pharmaceutical Care. It provides hospital-wide, pathogen-specific sensitivity patterns for major antibiotics at UIHC, cost and dosing information, parenteral to oral conversion information, and dosing with decreased renal function. It provides the clinician with readily available clinical data that allow for initial antibiotic selection based on hospital-wide sensitivity trends.

Due to the efforts of the Antibiotic Advisory Subcommittee and the Protocol Antibiotic Program, the susceptibility patterns at UIHC compare favorably with those of other major teaching hospitals. Only 17% of Staphylococcus aureus are resistant to methicillin - a level considerably lower than the community rate of 25%. Just 26% of Pseudomonas aeruginosa are resistant to gentamicin. Many other teaching hospitals no longer consider the use of gentamicin for Pseudomonas aeruginosa because their resistance rates are much higher. This is a significant achievement which is due to the ongoing efforts of UIHC staff to ensure the use of clinically appropriate therapy for the treatment of specific infections.

Appropriate Use of Drug Levels

Vancomycin
Vancomycin levels are frequently ordered inappropriately with uninterpretable results. Therefore, the AAS developed guidelines for the appropriate monitoring of levels. The guidelines were subsequently reviewed by the medical service chiefs and then approved by the P&T Subcommittee. The following guidelines were approved in October 1995, but improved adherence is still needed as many unnecessary levels are still being drawn. Following the guidelines more closely could lead to more appropriate dosing adjustments, as well as substantial laboratory savings.

WHO

WHO NOT

WHEN

HOW

Aminoglycosides
The results of serum aminoglycoside levels are often unusable because the levels are drawn incorrectly or at inappropriate times. This can result in suboptimal dosage adjustments. Uninterpretable levels can result in large amounts of wasted laboratory resources. There are two different methods of dosing aminoglycosides, and each has its own specific method for monitoring levels.

Multiple-Daily Dosed Aminoglycosides

HOW

WHEN

 

Extended Interval Dosing (EID) Aminoglycosides
Extended interval dosing of aminoglycosides can be useful in select patient populations. Traditional multiple daily dosing was designed to keep serum aminoglycoside concentrations above the minimum inhibitory concentration for most of the dosage interval, with the intent to prevent regrowth of organisms. High peaks were thought to correlate with toxicity, not improved antibacterial activity. Currently available data support the concept of administering larger doses less frequently. The rationale is based on the concentration-dependent bactericidal activity of aminoglycosides, the extended post-antibiotic effect, the possibility for reduced nephrotoxicity, and equivalent or reduced ototoxicity.

In vitro, the aminoglycosides eradicate bacteria at a rate proportional to the peak concentration attained. Therefore, high peak levels result in a more rapid and efficient bactericidal effect against susceptible organisms. In fact, peak aminoglycoside serum concentrations of 8 to12 times the minimum inhibitory concentration of the bacteria have been associated with a positive clinical outcome. The post-antibiotic effect (PAE) is defined as the time period that surviving bacteria, following exposure to an antibiotic, cannot metabolize or multiply even though extracellular antibiotic is no longer present. The duration of the PAE for aminoglycosides with gram negative bacteria has been reported to be from 3 to 24 hours in vivo, depending on the peak concentration and the organism. The prolonged post-antibiotic effect is another reason that extended interval dosing is a rational alternative.

Since the uptake of aminoglycosides into renal tubular cells is a saturable process, larger doses would not be expected to be any more nephrotoxic than smaller doses. Both animal and human studies have shown that the concentration in the renal cortex is significantly lower when administered as a single daily dose than when divided and administered more frequently. Animal data support an accumulation threshold in the organ of Corti as well, so there is a potential for less ototoxicity. Clinical trials consistently show that EID has equivalent or less toxicity than multiple daily dosing. Other advantages include a reduction in costs incurred by the institution for preparing, administering and monitoring therapy, and equal therapeutic effectiveness when compared with traditional dosing.

The Pharmacy and Therapeutics Subcommittee has authorized clinical pharmacy staff to determine the proper aminoglycoside dose and dosing interval and to coordinate serum level sampling to refine EID for aminoglycosides, upon request by a UIHC prescriber. If this service is desired, the prescriber should write "Extended-Interval Dosing for Gentamicin via Pharmacy" on a routine A-1a Doctors' Order form.

The following are guidelines for serum sampling when EID is used.

Summary
The Antibiotic Advisory Subcommittee is a multi-disciplinary group that looks at a number of issues regarding the appropriate use of antibiotics. Due to its efforts and the cooperation of the Medical and Pharmacy staff, UIHC has been successful at protecting the bacterial ecology. The appropriate use of antibiotic levels is another method by which medicine can be practiced more cost-effectively to make optimal use of limited resources.

Additional Information

Vancomycin Levels

Clin Infect Dis 1994;18:533-43.
Ann Pharmacother 1993;27:594-8.
Clin Infect Dis 1994;18:544-6.
J Antimicrob Chemother 1984;14SD:43-52.
Basic Clinical Pharmacokinetics, Third Edition. 1994; Pages 478-9.

Gentamicin Levels

J Infect Dis 1987; 155:93-9.
Am J Hosp Pharm 1978;35:317-20.
Basic Clinical Pharmacokinetics, Third Edition. 1994; Pages 136-8.
Antimicrob Agents Chemother 1982:21:407-11.

Aminoglycoside Extended-Interval Dosing

Clin Infect Dis 1997;24:796-809.
Clin Infect Dis 1997;24:786-95.
Clin Infect Dis 1997;24:810-15.
Antimicrob Agents Chemother 1995; 3:650-5.


PHARMACY AND THERAPEUTICS SUBCOMMITTEE ACTIONS

DRUGS ADDED TO STOCK

FENTANYL
Transmucosal Lozenge: 200 mcg, 400 mcg, 600 mcg
The transmucosal lozenge form of fentanyl (Actiq - Abbott) is indicated only for the management of breakthrough cancer pain in patients with malignancies who are already receiving and who are tolerant to opioid therapy for their underlying persistent cancer pain. Extensive patient/caregiver education is necessary to ensure proper storage and disposal of this product.

NOTE: Prescribing is restricted to attending staff physicians from Anesthesia and the Adult Hematology/Oncology Division.

ADDITIONAL ACTIONS

DELAVIRDINE (RESCRIPTOR") TABLETS

A 200 mg tablet was added to stock.

DIDANOSINE (VIDEX") CHEWABLE TABLET
A 200 mg chewable tablet was added to stock.

HYDROXYZINE TABLETS
A 50 mg tablet has been added to stock.

_______________________

Note: The cost following each brief monograph is the UIHC acquisition cost.

DRUGS DELETED FROM STOCK

ALUMINUM HYDROXIDE 600 MG (AMPHOGEL(R)) TABLETS Discontinued by the manufacturer. Aluminum hydroxide oral suspension and 400 mg oral capsules (Alu-Caps(R)) are available.

ALUMINUM HYDROXIDE WITH MAGNESIUM HYDROXIDE WITH SIMETHICONE (MAALOX(R) PLUS EXTRA STRENGTH) TABLETS Discontinued by the manufacturer. A suspension formulation is still available.

ATROPINE 0.5% OPHTHALMIC SOLUTION Discontinued by the manufacturer. Atropine 1% ophthalmic solution is available.

DANAZOL 50 MG TABLETS Deleted due to low use. A 200 mg tablet is available.

ISOSORBIDE (ISMOTIC(R)) ORAL SOLUTION Discontinued by the manufacturer. Glycerin oral solution is available.

NITROGLYCERIN 2% OINTMENT, 60 GRAM TUBE Deleted due to low use. A 30 gram size is still available.

PLASMA PROTEIN FRACTION (PPF) INJECTION Unavailable from any manufacturer. Albumin injection is available.

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